This book has been primarily design for the undergraduate, postgraduate and researchers in pharmaceutical chemistry. In a broader perspective, the students studying pharmaceutical sciences at undergraduate, postgraduate or researchers shall be grossly benefited by it’s well planned, systematically developed, structured, illustrated, expanded and elaborated subject matter. It contains all the basic concepts and principles that a researcher should know about the different aspects of the synthesis including the biological activity of the pharmaceutical compounds. This book also provides spectral analysis of newly synthesize compounds. The book is well illustrated. Hopefully it will serve as a key to the undergraduate, postgraduate and researchers in pharmaceutical chemistry.The authors earnestly believe that the wide coverage various synthetic schemes would certainly render pharmaceutical chemistry to serve as an exclusive source of information’s, ideas, inspiration towards research and finding newer possible practical solutions to problems encountered in the synthesis of pharmaceutical compounds.